The first and simple total synthesis of cappariloside A1

The first and simple total synthesis of cappariloside A1

フォーマット:

論文

責任表示:

Somei, Masanori ; Yamada, Fumio

言語:

英語

出版情報:

日本複素環化学研究所, 2000-07-01

著者名:

掲載情報:

Heterocycles

巻:

53

通号:

7

開始ページ:

1573

終了ページ:

1578

バージョン:

publisher

概要:

金沢大学大学院自然科学研究科生理活性物質科学<br />金沢大学薬学部<br />A lithium hydroxide promoted simple glycosylation of 4-hydroxyindole-3- acetonitrile with 2,3,4, 6-tetra-O-acetyl-a-D-glucopyranosyl bromide was developed. Utilizing the method, the first and five steps total synthesis of cappariloside A was achieved from indole-3-carbaldehyde in 41% overall yield.

URL:

http://hdl.handle.net/2297/4360

タイトル・著者・出版者が同じ資料

詳細

主題:	cappariloside a; drug synthesis
受理日:	2000-07-01

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