Nucleophilic substitution reaction on the nitrogen of indole nucleus: Formation of 1-(indol-3-yl)indoles upon reaction of 1-hydroxyindoles with indole in formic acid

Nucleophilic substitution reaction on the nitrogen of indole nucleus: Formation of 1-(indol-3-yl)indoles upon reaction of 1-hydroxyindoles with indole in formic acid

フォーマット:

論文

責任表示:

Somei, Masanori ; Yamada, Fumio ; Hayashi, Toshikatsu ; Goto, Aya ; Saga, Yoshitomo

言語:

英語

出版情報:

日本複素環化学研究所, 2001-03-01

著者名:

掲載情報:

Heterocycles

巻:

55

通号:

3

開始ページ:

457

終了ページ:

460

バージョン:

publisher

概要:

金沢大学大学院自然科学研究科生理活性物質科学<br />金沢大学薬学部<br />1-(Indol-3-yl)indoles are obtained in excellent to good yields by the reaction of 1-hydroxyindoles with indole in 85% formic acid. Their structures are determined by X-Ray crystallographic analysis and chemical correlations. The unprecidented SN2 mechanism on the indole nitrogen is proposed.

URL:

http://hdl.handle.net/2297/4366

タイトル・著者・出版者が同じ資料

詳細

主題:	1 (indol 3 yl)indole derivative; 1 hydroxyindole derivative; indole derivative; nitrogen
受理日:	2001-03-01

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