A novel preparation of 3-hydroxy-3H-indole-3-ethanamines and -3H-indole-3-acetamides having either a 4-morpholinyl or 1-pyrrolidinyl group at the 2-position

A novel preparation of 3-hydroxy-3H-indole-3-ethanamines and -3H-indole-3-acetamides having either a 4-morpholinyl or 1-pyrrolidinyl group at the 2-position

フォーマット:

論文

責任表示:

Hayashi, Toshikatsu ; Nakai, Yu-ya ; Yamada, Fumio ; Somei, Masanori

言語:

英語

出版情報:

日本複素環化学研究所, 2004-01-01

著者名:

掲載情報:

Heterocycles

巻:

62

開始ページ:

437

終了ページ:

444

バージョン:

publisher

概要:

金沢大学大学院自然科学研究科生理活性物質科学<br />金沢大学薬学部<br />A novel synthetic method is discovered for 3-hydroxy-3H-indole-3-ethanamines and -3H-indole-3-acetamides having either a 4-morpholinyl or 1-pyrrolidinyl group at the 2-position by reacting the corresponding 1-hydroxyindoles with enamines in the presence of tosyl or mesyl chloride. A plausible mechanism is proposed.

URL:

http://hdl.handle.net/2297/4379

タイトル・著者・出版者が同じ資料

詳細

主題:	3 hydroxy 3h indole 3 ethanamine derivative; acetamide derivative; ethylamine; hydroxy 3h indole 3 acetamide derivative derivative; indole; morpholine derivative
受理日:	2004-01-01

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