Short step synthesis of an antibiotic, 6-cyano-5-methoxy-12-methylindolo[2,3-a]carbazole

Short step synthesis of an antibiotic, 6-cyano-5-methoxy-12-methylindolo[2,3-a]carbazole

フォーマット:

論文

責任表示:

Somei, Masanori ; Yamada, Fumio ; Suzuki, Yoshiaki ; Ohmoto, Shinobu ; Hayashi, Hiroyuki

言語:

英語

出版情報:

日本複素環化学研究所, 2004-12-31

著者名:

掲載情報:

Heterocycles

巻:

64

開始ページ:

483

終了ページ:

489

バージョン:

publisher

概要:

金沢大学大学院自然科学研究科生理活性物質科学<br />For evaluating the effectiveness of organic synthesis, both intellectual property factor (IPF) and application potential factor (APF) are proposed. As a representative example, a highly effective synthetic … method with IPF value of 53.8 and APF value of 100 has been established starting from indigo directing toward an antibiotic, 6-cyano-5-methoxy-12-methylindolo[2,3-a]carbazole, using only conventional reagents without using any protecting groups. © 2004 The Japan Institute of Heterocyclic Chemistry All rights reserved. 続きを見る

URL:

http://hdl.handle.net/2297/4381

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受理日:	2004-12-31

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4 論文 Simple synthesisi of 2-2'-bisindole from indigo and its application for the syntheses of indole[2,3-a]pyrrolo[3,4-c]carbazole-5,7-(6H9dione and -5-(6H9one … Somei, Masanori, Hayashi, Hiroyuki, Izumi, Tohru, Ohmoto, Shinobu 日本複素環化学研究所	10 論文 Nucleophilic Substitution Reaction in Indole Chemistry: 1-Methoxy-6-nitroindole-3-carbaldehyde as a Versatile Building Block for 2,3,6-Trisubstituted Indoles Yamada, Koji, Yamada, Fumio, Shiraishi, Takei, Tomioka, Saori, Somei, Masanori Japan Institute of Heterocyclic Chemistry = 日本複素環化学研究所
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